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Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T5319 |
Rimeporide
EMD-87580 |
Sodium Channel | Membrane transporter/Ion channel |
Rimeporide (EMD-87580) 是有效的 Na+/H+交换泵 (NHE-1) 选择性抑制剂。 | |||
T2238 |
Cariporide
卡立泊来德,HOE-642 |
Sodium Channel | Membrane transporter/Ion channel |
Cariporide (HOE-642) 是一种选择性的Na+/H+交换抑制剂。 | |||
T5333 |
Rimeporide hydrochloride
盐酸Rimeporide,EMD-87580 hydrochloride |
Sodium Channel | Membrane transporter/Ion channel |
Rimeporide hydrochloride (EMD-87580 hydrochloride) 是一种有效的 Na+/H+交换泵(NHE-1) 选择性抑制剂。 | |||
T7587 |
Tenapanor
RDX-5791,RDX 5791,AZD 1722,Tenapanor free base,RDX5791,AZD-1722,AZD1722 |
Sodium Channel | Membrane transporter/Ion channel |
Tenapanor (RDX 5791) 是钠氢离子交换NHE3的有效抑制剂, 对人和大鼠NHE3的IC50分别是5和10 nM。 | |||
TQ0157 |
EIPA
L593754,MH 12-43 |
Sodium Channel; TRP/TRPV Channel | Membrane transporter/Ion channel |
EIPA (L593754) 是一种有效的TRPP3 channel 抑制剂,IC50为 10.5 μM。EIPA 对Na+/H+交换 (NHE) 和巨噬细胞也有抑制作用。 | |||
T12219 |
NHE3-IN-1
|
Sodium Channel | Membrane transporter/Ion channel |
NHE3-IN-1 是钠/质子交换剂 3 (NHE-3) 的抑制剂。 | |||
T11172 |
EIPA hydrochloride
L593754 hydrochloride,MH 12-43 hydrochloride |
TRP/TRPV Channel | Membrane transporter/Ion channel |
EIPA hydrochloride also inhibits Na+/H+-exchanger (NHE) and macropinocytosisEIPA hydrochloride (L593754 hydrochloride) is a TRPP3 channel inhibitor with an IC50 of 10.5 μM. |
Cat. No. | Product Name | Target | Signaling Pathways |
---|---|---|---|
T1033 |
Monensin sodium salt
莫能菌素钠盐,Sodium Monensin,Monensin A sodium salt |
Sodium Channel; Antibacterial; Antibiotic | Membrane transporter/Ion channel; Microbiology/Virology |
Monensin sodium salt (Monensin A sodium salt) 是由肉桂链霉菌 分泌的抗生素。它是一种介导Na+/H+交换的离子载体。它引起细胞多泡体 (MVBs) 增大并调节外泌体的分泌。 |